Tirabrutinib, CAS 1351636-18-4

Tirabrutinib, CAS 1351636-18-4
Artikelnummer
TGMTQ0236-200mg
Verpackungseinheit
200 mg
Hersteller
TargetMol Chemicals

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Description: Tirabrutinib (GS-4059) (ONO-4059) is an orally active Bruton’s Tyrosine Kinase (Btk) inhibitor (can cross the blood-brain barrier (BBB)), with an IC50 of 6.8 nM. Tirabrutinib irreversibly and covalently binds to Btk and inhibits aberrant B cell receptor signaling. Tirabrutinib can be used in studies of autoimmune diseases and hematological malignancies.

CAS Number: 1351636-18-4

Formula: C25H22N6O3

Molecular Weight: 454,48

References: Dhillon S. Tirabrutinib: First Approval. Drugs. 2020 Jun;80(8):835-840.
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Artikelnummer TGMTQ0236-200mg
Hersteller TargetMol Chemicals
Hersteller Artikelnummer TQ0236-200mg
Verpackungseinheit 200 mg
Mengeneinheit STK
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