Product Description: Sulfo-PDBA-DM4 is a agent-linker conjugate composed of a potent a tubulin inhibitor DM4 and a linker Sulfo-PDBA to make antibody agent conjugate (ADC). Sulfo-PDBA is a gluthatione cleavable linker.
Applications: COVID-19-immunoregulation
Formula: C42H60ClN3O15S3
References: [1]Sun X, et al. Effects of Drug-Antibody Ratio on Pharmacokinetics, Biodistribution, Efficacy, and Tolerability of Antibody-Maytansinoid Conjugates. Bioconjug Chem. 2017 May 17;28(5):1371-1381.
CAS Number: 1461704-01-7
Molecular Weight: 978.58
Research Area: Cancer; Inflammation/Immunology
Solubility: 10 mM in DMSO
Target: Drug-Linker Conjugates for ADC