Fenvalerate-d5, CAS 1246815-00-8

Product Description: Fenvalerate-d5 is the deuterium labeled Fenvalerate. Fenvalerate is a potent protein phosphatase 2B (calcineurin) inhibitor with an IC50 of 2-4 nM for PP2B-Aα. Fenvalerate is a pyrethroid ester insecticide and acaricide[1].

Formula: C25H17D5ClNO3

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216. /[2]E Enan, et al. Specific Inhibition of Calcineurin by Type II Synthetic Pyrethroid Insecticides. Biochem Pharmacol. 1992 Apr 15;43(8):1777-84.;A R Reilein, et al. Regulation of Organelle Movement in Melanophores by Protein Kinase A (PKA), Protein Kinase C (PKC), and Protein Phosphatase 2A (PP2A). J Cell Biol. 1998 Aug 10;142(3):803-13.

CAS Number: 1246815-00-8

Molecular Weight: 424.93

Research Area: Infection

Solubility: 10 mM in DMSO

Target: Bacterial;Isotope-Labeled Compounds;Phosphatase

• Artikelnummer: MEXHY-B2006S-2500UG
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-B2006S-2500UG
• Green Labware: Nein
• Verpackungseinheit: 2500 ug
• Mengeneinheit: STK