Tebuconazole-d9, CAS 1246818-83-6

Product Description: Tebuconazole-d9 is the deuterium labeled Tebuconazole. Tebuconazole is an agricultural azole fungicide which can also inhibit CYP51 with IC50s of 0.9 and 1.3 μM for Candida albicans CYP51 (CaCYP51) and truncated Homo sapiens CYP51 (Δ60HsCYP51), respectively.

Formula: C16H13D9ClN3O

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216. /[2]Warrilow AG, et al. Azole affinity of sterol 14α-demethylase (CYP51) enzymes from Candida albicans and Homo sapiens. Antimicrob Agents Chemother. 2013 Mar;57(3):1352-60.

CAS Number: 1246818-83-6

Molecular Weight: 316.87

Research Area: Infection

Solubility: 10 mM in DMSO

Target: Cytochrome P450;Fungal

• Artikelnummer: MEXHY-B0852S-1
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-B0852S-1
• Green Labware: Nein
• Verpackungseinheit: 1 mg
• Mengeneinheit: STK