Amauromine, CAS 88360-87-6

Formulation: A solid

Formal Name: (5aS,7aS,8aR,13aS,15aS,16aR)-8a,16a-bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-pyrazino[1'',2'':1,5;4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione

Purity: ≥98%

Formula Markup: C32H36N4O2

Formula Weight: 508,7

Shelf life (days): 1460

CAS Number: 88360-87-6

Notes: Amauromine is a neutral antagonist of the cannabinoid (CB) receptor CB1 that is selective for CB1 (Ki = 178 nM; Kb = 66.6 nM) over CB2, with no activity at CB2 receptors at concentrations up to 10 µM.{36266} It is also an antagonist of GPR18 (IC50 = 3.74 µM).{36265} Amauromine has vasodilatory activity.{36267}

• Artikelnummer: CAY23886-1
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 23886-1
• Green Labware: Nein
• Verpackungseinheit: 1 mg
• Mengeneinheit: STK