Formulation: A powder
Formal Name: N2-(1,9-dioxo-10,12-octadecadien-1-yl)-D-glutaminyl-L-threonyl-β-alanyl-D-tryptophyl-D-seryl-glycine, (6→2)-lactone
Purity: ≥95%
Formula Markup: C46H66N8O11
Formula Weight: 907,1
Shelf life (days): 1460
CAS Number: 156223-08-4
Notes: Aselacin C is a cyclic pentapeptolide antagonist of endothelin receptor type A (ETA) and ETB originally isolated from Acremonium.{61234} It inhibits the binding of endothelin-1 to isolated bovine atrial membranes and porcine cerebral membranes, which endogenously express high levels of ETA and ETB, respectively, with IC50 values of 60 and 80 µg/ml, respectively.