Bilaid C, CAS 2393866-13-0

Formulation: A solid

Formal Name: L-tyrosyl-D-valyl-L-valyl-D-phenylalanine

Purity: ≥95%

Formula Markup: C28H38N4O6

Formula Weight: 526,6

Shelf life (days): 1460

CAS Number: 2393866-13-0

Notes: Bilaid C is a tetrapeptide µ-opioid receptor agonist (Ki = 210 nM in HEK293 cell membranes expressing the human receptor) that has been found in Penicillium.{57195} It inhibits forskolin-induced cAMP accumulation by 77% in HEK293 cells expressing the human µ-opioid receptor when used at a concentration of 10 µM. Bilaid C induces inward rectifying potassium channel (Kir) currents in rat locus coeruleus slices that endogenously express high levels of the µ-opioid receptor (EC50 = 4.2 µM).

• Artikelnummer: CAY31246-1
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 31246-1
• Green Labware: Nein
• Verpackungseinheit: 1 mg
• Mengeneinheit: STK