BRL 15572, CAS 193611-72-2

Formulation: A solid

Formal Name: 4-(3-chlorophenyl)-α-(diphenymethyl)-1-piperazineethanol, dihydrochloride

Purity: ≥98%

Formula Markup: C25H27ClN2O • 2HCl

Formula Weight: 479,9

Shelf life (days): 1460

CAS Number: 193611-72-2

Notes: BRL 15572 is an antagonist of the serotonin (5-HT) receptor subtype 5-HT1D (Ki = 0.013 µM in CHO cell membranes expressing the human receptor).{54405} It is selective for 5-HT1D over several other G protein-coupled 5-HT receptor subtypes with Ki values ranging from 0.25 to 6.3 µM but does bind 5-HT1A and 5-HT2B receptors (Kis = 0.02 and 0.04 µM, respectively). BRL 15572 also acts as a partial agonist at 5-HT1D receptors (EC50 = 0.008 µM in a [35S]GTPγS binding assay).

• Artikelnummer: CAY31191-100
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 31191-100
• Green Labware: Nein
• Verpackungseinheit: 100 mg
• Mengeneinheit: STK