BRL 54443, CAS 57477-39-1

Formulation: A crystalline solid

Formal Name: 3-(1-methyl-4-piperidinyl)-1H-indol-5-ol

Purity: ≥98%

Formula Markup: C14H18N2O

Formula Weight: 230,3

Shelf life (days): 1460

CAS Number: 57477-39-1

Notes: BRL 54443 is a potent agonist of the serotonin (5-HT) receptor subtypes 5-HT1E and 5-HT1F (Ki values are 1.1 and 0.7 nM, respectively).{33346} It displays more than 30-fold selectivity over other 5-HT and dopamine receptors. At higher concentrations, BRL 54443 induces 5-HT2A-mediated contraction of mouse thoracic aorta strips in vitro (pEC50 = 6.5).{33347} It significantly reduces formalin-induced pain in rat hind paw.{33345}

• Artikelnummer: CAY21263-5
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 21263-5
• Green Labware: Nein
• Verpackungseinheit: 5 mg
• Mengeneinheit: STK