Carteolol (hydrochloride), CAS 51781-21-6

Formulation: A crystalline solid

Formal Name: 5-[3-[(1,1-dimethylethyl)amino]-2-hydroxypropoxy]-3,4-dihydro-2(1H)-quinolinone, monohydrochloride

Purity: ≥98%

Formula Markup: C16H24N2O3 • HCl

Formula Weight: 328,8

Shelf life (days): 1460

CAS Number: 51781-21-6

Notes: Carteolol is an antagonist of β-adrenergic receptors (Kd = 13 nM).{38754,38755} It blocks isoproterenol-induced increases in heart rate, contractile force, and blood pressure in vagotomized dogs (ED50s = 2.3, 3.1, and 1.8 µg/kg, respectively).{38756} The (R) and (S)-enantiomers of carteolol reduce intraocular pressure to similar levels in rabbits when applied topically as a 1% solution.{38757} Formulations containing carteolol have been used in the treatment of open-angle glaucoma.

• Artikelnummer: CAY23758-100
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 23758-100
• Green Labware: Nein
• Verpackungseinheit: 100 mg
• Mengeneinheit: STK