Formulation: A solid
Formal Name: 3-(2,5-difluorophenyl)-7-[1,1-di(methyl-d3)ethyl-2,2,2-d3]-6-[(1-methyl-1H-1,2,4-triazol-5-yl)methoxy]-1,2,4-triazolo[4,3-b]pyridazine
Purity: ≥99% (deutereated forms d1-d9)
Formula Markup: C19H10D9F2N7O
Formula Weight: 408,5
Shelf life (days): 1460
CAS Number: 1213669-91-0
Notes: CTP354 is a deuterated derivative of the GABAA receptor modulator L-838,417.{67059} It binds to the GABAA receptor benzodiazepine binding site in non-α1 subunit-containing GABAA receptors. CTP354 has a longer duration of action than L-838,417 in a rat model of neuropathic pain induced by sciatic nerve ligation.