CYM 2503, CAS 1308833-36-4

Formulation: A solid

Formal Name: 3-cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanyl-N-(1,2-dihydro-4-methyl-2-oxo-7-quinolinyl)-N6-[(1,1-dimethylethoxy)carbonyl]-L-lysinamide

Purity: ≥95%

Formula Markup: C45H55N5O7

Formula Weight: 778

Shelf life (days): 1460

CAS Number: 1308833-36-4

Notes: CYM 2503 is a positive allosteric modulator (PAM) of the galanin-2 (GAL2) receptor.{64502} It enhances the production of inositol monophosphate (IP1) induced by galanin in HEK293 cells expressing the GAL2 receptor (EC50 = 0.69 µM). CYM 2503 (60 mg/kg) increases the latency to first electrographic and behavioral seizures and reduces mortality in a lithium-pilocarpine (Li-pilocarpine) rat model of status epilepticus.

• Artikelnummer: CAY36590-10
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 36590-10
• Green Labware: Nein
• Verpackungseinheit: 10 mg
• Mengeneinheit: STK
• Methode: Reinstoffe