Mirogabalin, CAS 1138245-13-2

Formulation: A crystalline solid

Formal Name: (1R,5S,6S)-6-(aminomethyl)-3-ethyl-bicyclo[3.2.0]hept-3-ene-6-acetic acid

Purity: ≥98%

Formula Markup: C12H19NO2

Formula Weight: 209,3

Shelf life (days): 1460

CAS Number: 1138245-13-2

Notes: Mirogabalin is a calcium channel blocker with analgesic effects.{36068} It binds to the α2δ-1 and α2δ-2 subunits of voltage-dependent Ca2+ channels. Mirogabalin has potent and sustained analgesic effects (ED50 = 2.5 mg/kg) in rats with diabetes induced by streptozotocin (STZ; Item No. 13104). Mirogabalin does not inhibit activities associated with CNS adverse effects of analgesics, such as rotarod performance (ID50 = 9.4 mg/kg) or locomotor activity (ID50 = 43.9 mg/kg), at its effective dose.

• Artikelnummer: CAY22475-1
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 22475-1
• Green Labware: Nein
• Verpackungseinheit: 1 mg
• Mengeneinheit: STK