Nemonapride, CAS 75272-39-8

Formulation: A crystalline solid

Formal Name: rel-5-chloro-2-methoxy-4-(methylamino)-N-[(2R,3R)-2-methyl-1-(phenylmethyl)-3-pyrrolidinyl]-benzamide

Purity: ≥98%

Formula Markup: C21H26ClN3O2

Formula Weight: 387,9

Shelf life (days): 1460

CAS Number: 75272-39-8

Notes: Nemonapride is an antipsychotic that readily passes through the blood brain barrier and exhibits potent neuroleptic effects in animals.{34046} It binds dopamine 2 (D2)-like receptors preferentially over D1-like receptors (Kis = 0.06, 0.3, and 0.15 nM for D2, D3, and D4, respectively).{34046,32473} Nemonapride also binds sigma 1 (σ1) and σ2 receptors (Kis = 8.4 and 9.6 nM, respectively) and activates the serotonin 1A receptor (5-HT1A; IC50 = 34 nM).{34047,34045}

• Artikelnummer: CAY21376-1
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 21376-1
• Green Labware: Nein
• Verpackungseinheit: 1 mg
• Mengeneinheit: STK