Olodaterol, CAS 868049-49-4

Formulation: A crystalline solid

Formal Name: 6-hydroxy-8-[(1R)-1-hydroxy-2-[[2-(4-methoxyphenyl)-1,1-dimethylethyl]amino]ethyl]-2H-1,4-benzoxazin-3(4H)-one

Purity: ≥98%

Formula Markup: C21H26N2O5

Formula Weight: 386,4

Shelf life (days): 1460

CAS Number: 868049-49-4

Notes: Olodaterol is a selective agonist of β2-adrenergic receptors (β2-ARs; EC50s = 97.7 and 2,725 nM for human β2- and β1-ARs, respectively).{40022} In vivo, olodaterol completely reverses acetylcholine-induced bronchoconstriction without cardiovascular side effects in guinea pigs. It also exhibits dose-dependent bronchoprotection in a beagle model of acetylcholine-induced bronchoconstriction for a period of 24 hours, indicating potential for once-daily dosing.{40023} Formulations containing olodaterol have been used to treat bronchoconstriction associated with chronic obstructive pulmonary disease.{40024}

• Artikelnummer: CAY21794-10
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 21794-10
• Green Labware: Nein
• Verpackungseinheit: 10 mg
• Mengeneinheit: STK