Raloxifene 6-Glucuronide, CAS 174264-50-7

Formulation: A solid

Formal Name: 2-(4-hydroxyphenyl)-3-[4-[2-(1-piperidinyl)ethoxy]benzoyl]benzo[b]thien-6-yl, β-D-glucopyranosiduronic acid

Purity: ≥90%

Formula Markup: C34H35NO10S

Formula Weight: 649,7

Shelf life (days): 1460

CAS Number: 174264-50-7

Notes: Raloxifene 6-glucuronide is a metabolite of the selective estrogen receptor modulator raloxifene (Item No. 10011620).{42731} It is formed from raloxifene via the UDP-glucuronosyltransferase (UGT) isoforms UGT1A1 and UGT1A8. It binds to the estrogen receptor with an IC50 value of 290 nM.{42731,42732} Unlike raloxifene, raloxifene 6-glucuronide does not inhibit the voltage-gated potassium channel Kv4.3.{42733}

• Artikelnummer: CAY27832
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 27832-1
• Green Labware: Nein
• Verpackungseinheit: 1 mg
• Mengeneinheit: STK