Tolperisone-d10 (hydrochloride), CAS 1185160-65-9

Formulation: A solid

Formal Name: 3-2,2,3,3,4,4,5,5,6,6-decadeuteriopiperidin-1-yl)-2-methyl-1-(4-methylphenyl)propan-1-one, monohydrochloride)

Purity: ≥99% deuterated forms (d1-d10)

Formula Markup: C16H13D10NO • HCl

Formula Weight: 291,9

Shelf life (days): 1460

CAS Number: 1185160-65-9

Notes: Tolperisone-d10 is intended for use as an internal standard for the quantification of tolperisone by GC- or LC-MS. Tolperisone is a piperidine that acts as an inhibitor of voltage-gated sodium channels with an IC50 value of 198 µM, for inhibition of peak sodium currents evoked by step depolarizations in dorsal root ganglion (DRG) neurons, in vitro.{34788} Tolperisone acts as an antispastic agent that attenuates monosynaptic, disynaptic, and polysynaptic reflux response to dorsal root stimulation in vivo. Formulations containing tolperisone are used as analgesics and muscle relaxants.

• Artikelnummer: CAY22592-1
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 22592-1
• Green Labware: Nein
• Verpackungseinheit: 1 mg
• Mengeneinheit: STK
• Methode: GC-MS, LC-MS, Isotopenmarkierung