Product Description: Axelopran (TD-1211) is an opioid receptor antagonist with pKi values of 9.8, 8.8 and 9.9 for human recombinant μ and δ receptors and guinea pig κ receptor, respectively.
Applications: Neuroscience-Neuromodulation
Formula: C26H39N3O4
References: [1]Tsuruda PR, et al., The in vitro pharmacological profile of TD-1211, a neutral opioid receptor antagonist. Naunyn Schmiedebergs Arch Pharmacol. 2013 Jun;386(6):479-91.
CAS Number: 949904-48-7
Molecular Weight: 457.61
Research Area: Neurological Disease
Target: Opioid Receptor