Product Description: Cetrorelix Acetate (SB-75 acetate) is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM[1].
Applications: Neuroscience-Neuromodulation
Formula: C72H96ClN17O16
References: [1]Beckers T et al. Characterization of gonadotropin-releasing hormone analogs based on a sensitive cellular luciferase reporter gene assay. Anal Biochem. 1997 Aug 15;251(1):17-23./[2]Gründker C et al. Role of gonadotropin-releasing hormone (GnRH) in ovarian cancer. Reprod Biol Endocrinol. 2003 Oct 7;1:65.
CAS Number: 145672-81-7
Molecular Weight: 1491.09
Compound Purity: 99.87
Research Area: Neurological Disease; Endocrinology