GLP-1R/GIPR agonist-1 (soduim)

Product Description: GLP-1R/GIPR agonist-1 soduim is the sodium salt form of GLP-1R/GIPR agonist-1 (HY-P10302). GLP-1R/GIPR agonist-1 soduim is a dual agonist for glucagon-like peptide-1 receptor (GLP-1R, EC50 is 0.57 nM) and glucose-dependent insulin releasing peptide receptor (GIPR, EC50 is 0.75 nM). GLP-1R/GIPR agonist-1 soduim lowers blood sugar by mimicking the action of endogenous hormones GLP-1 and GIP, enhancing insulin secretion while inhibiting glucagon secretion. GLP-1R/GIPR agonist-1 soduim can be used in the study of metabolic diseases such as diabetes, obesity, and non-alcoholic steatohepatitis (NASH)[1].

Applications: Metabolism-sugar/lipid metabolism

Formula: C220H342N55O69.xNa

References: [1]Liu C, et al. Discovery of a novel GLP-1/GIP dual receptor agonist CY-5 as long-acting hypoglycemic, anti-obesity agent[J]. Bioorganic Chemistry, 2021, 106: 104492.

Molecular Weight: 4861.38 (free base)

Compound Purity: 96.55

Research Area: Metabolic Disease

Target: GLP Receptor

• Artikelnummer: MEXHY-P10302A-5
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-P10302A-5
• Green Labware: Nein
• Verpackungseinheit: 5 mg
• Mengeneinheit: STK