Formulation: A solid
Formal Name: 2-[(6-benzo[b]thien-2-ylthieno[3,2-d]pyrimidin-4-yl)thio]-acetic acid
Purity: ≥98%
Formula Markup: C16H10N2O2S3
Formula Weight: 358,5
Shelf life (days): 1460
CAS Number: 2650530-00-8
Notes: SGC-STK17B-1 is an inhibitor of serine/threonine kinase 17b (STK17B), also known as DRAK2 (IC50 = 43 nM).{69792} It is selective for STK17B over STK17A (IC50 = 4,700 nM), as well as eight additional kinases (IC50s = 5,200->10,000 nM). See the Structural Genomics Consortium (SGC) website for more information.