Entacapone, CAS 130929-57-6

Products from BPS Bioscience require a minimum order value above 400€

Biological Activity: Entacapone potently inhibits rat liver total COMT with IC50 and Ki values of 20.1 nM and 10.7 nM respectively. The IC50 values of entacapone against rat liver soluble COMT (S-COMT) and rat liver membrane-bound COMT (MB-COMT) are 14.3 nM and 73.3 nM respectively.

CAS Number: 130929-57-6

Description: Entacapone is a second-generation catechol-O-methyltransferase (COMT) inhibitor

Purity: ≥98% by HPLC

Solubility: Soluble in DMSO 61 mg/ml, water <1 mg/ml, ethanol 2 mg/ml

Storage Stability: Store at or below -20°C. Solid form is stable at least 12 months from date of receipt, when stored as directed. Do not store aqueous solutions for more than one day.

Target: COMT

Biosafety Level: Not applicable (BSL-1)

References: Forsberg M, et al. J Pharmacol Exp Ther. 2003 Feb;304(2):498-506.

• Artikelnummer: BPS27621-1
• Hersteller: BPS Bioscience
• Hersteller Artikelnummer: 27621-1
• Green Labware: Nein
• Verpackungseinheit: 10 mg
• Mengeneinheit: STK