Formulation: A solid
Formal Name: N-[5-[3-(3-hydroxy-1-piperidinyl)-1,2,4-oxadiazol-5-yl]-4-methyl-2-thiazolyl]-acetamide
Purity: ≥98%
Formula Markup: C13H17N5O3S
Formula Weight: 323,4
Shelf life (days): 1460
CAS Number: 1292300-75-4
Notes: TASP0415914 is a PI3Kγ inhibitor (IC50 = 29 nM).{51799} It is selective for PI3Kγ over Akt (IC50 = 294 nM). In vivo, TASP0415914 (30 and 100 mg/kg) reduces ankle redness and swelling in a mouse model of collagen-induced arthritis.