Androgen receptor-IN-3, CAS 926228-58-2

Androgen receptor-IN-3, CAS 926228-58-2
Artikelnummer
MEXHY-131953-0
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MedChemExpress

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Product Description: Androgen receptor-IN-3 (Compound 22) is an androgen receptor inhibitor. Androgen receptor-IN-3 inhibits AR-driven transcriptional activity in LNCaP cells, with an IC50 of 5.04 μM[1].

Formula: C14H16N2O2S

References: [1]Li H, et al. Discovery of small-molecule inhibitors selectively targeting the DNA-binding domain of the human androgen receptor. J Med Chem. 2014 Aug 14;57(15):6458-67.

CAS Number: 926228-58-2

Molecular Weight: 276.35

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Androgen Receptor
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Artikelnummer MEXHY-131953-0
Hersteller MedChemExpress
Hersteller Artikelnummer HY-131953-0
Green Labware Nein
Verpackungseinheit Get quote
Mengeneinheit STK
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