Antitumor agent-150

Antitumor agent-150
Artikelnummer
MEXHY-162450-0
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MedChemExpress

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Product Description: Antitumor agent-150 (V10), an anti-breast cancer agent, is a PROTAC-based MDM2 protein degrader (Red: Ganoderic acid A; Black: 4O-PEG linker; Blue: VHL ligand)[1].

Applications: Cancer-programmed cell death

Formula: C70H106N8O14S

References: [1]Yan Li, et al. Discovery of ganoderic acid A (GAA) PROTACs as MDM2 protein degraders for the treatment of breast cancer. Eur J Med Chem. 2024 Apr 15:270:116367.

Molecular Weight: 1315.70

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Apoptosis;MDM-2/p53;PROTACs
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Artikelnummer MEXHY-162450-0
Hersteller MedChemExpress
Hersteller Artikelnummer HY-162450-0
Green Labware Nein
Verpackungseinheit Get quote
Mengeneinheit STK
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