EZH2-IN-16, CAS 2238820-26-1

Product Description: EZH2-IN-16 (Compound 24) is an inhibitor for histone methyltransferase (EZH2). EZH2-IN-16 inhibits EZH2 and EZH2 Y641F, with IC50 of 37.6 and 79.1 nM. EZH2-IN-16 inhibits proliferation of WSU-DLCL2, with GI50 of 0.2 μM[1].

Formula: C32H38N4O4

References: [1]Zhou B, et al., Discovery of IHMT-EZH2-115 as a Potent and Selective Enhancer of Zeste Homolog 2 (EZH2) Inhibitor for the Treatment of B-Cell Lymphomas. J Med Chem. 2021 Oct 28;64(20):15170-15188.

CAS Number: 2238820-26-1

Molecular Weight: 542.67

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Histone Methyltransferase

• Artikelnummer: MEXHY-149463-0
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-149463-0
• Green Labware: Nein
• Verpackungseinheit: Get quote
• Mengeneinheit: STK