Description: GW9662 (TIMTEC-BB SBB006523) is a specific PPARγ antagonist (IC50: 3.3 nM, in a cell-free assay), with 100 to 1000-fold functional selectivity for PPARγ than PPARα/δ in cells.
CAS Number: 22978-25-2
Formula: C13H9ClN2O3
Molecular Weight: 276,68
References: Leesnitzer LM, et al. Biochemistry, 2002, 41(21), 6640-6650.