KSL 128114, CAS 2757292-12-7

KSL 128114, CAS 2757292-12-7
Artikelnummer
MEXHY-P10331-0
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MedChemExpress

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Product Description: KSL 128114, a peptide inhibitor of syntenin, binds the PDZ1 domain of syntenin with nanomolar affinity. KSL 128114 is resistant toward degradation in human plasma and mouse hepatic microsomes and displays a global PDZ domain selectivity for syntenin[1].

Formula: C96H165N39O21

References: [1]Linda M Haugaard-Kedström, et al. A High-Affinity Peptide Ligand Targeting Syntenin Inhibits Glioblastoma. J Med Chem. 2021 Feb 11;64(3):1423-1434.

CAS Number: 2757292-12-7

Molecular Weight: 2201.59

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Others
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Artikelnummer MEXHY-P10331-0
Hersteller MedChemExpress
Hersteller Artikelnummer HY-P10331-0
Green Labware Nein
Verpackungseinheit Get quote
Mengeneinheit STK
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