KYP-2047, CAS 796874-99-2

Product Description: KYP-2047 is a potent and BBB-penetrating prolyl-oligopeptidase (POP) inhibitor, with an Ki value of 0.023 nM. KYP-2047 reduces glioblastoma proliferation through angiogenesis and apoptosis modulation[1][2].

Applications: Cancer-programmed cell death

Formula: C20H25N3O2

References: [1]Jalkanen AJ, et al. Beneficial effect of prolyl oligopeptidase inhibition on spatial memory in young but not in old scopolamine-treated rats. Basic Clin Pharmacol Toxicol. 2007 Feb;100(2):132-8./[2]Scuderi SA, et al. KYP-2047, an Inhibitor of Prolyl-Oligopeptidase, Reduces GlioBlastoma Proliferation through Angiogenesis and Apoptosis Modulation. Cancers (Basel). 2021 Jul 9;13(14):3444.

CAS Number: 796874-99-2

Molecular Weight: 339.43

Compound Purity: 99.68

Research Area: Cancer

Solubility: DMSO : 100 mg/mL (ultrasonic)

Target: Apoptosis;MDM-2/p53;Prolyl Endopeptidase (PREP)

• Artikelnummer: MEXHY-100475-10.1
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-100475-10.1
• Green Labware: Nein
• Verpackungseinheit: 10mM/1mL
• Mengeneinheit: STK