PAD4-IN-2, CAS 2642327-52-2

PAD4-IN-2, CAS 2642327-52-2
Artikelnummer
MEXHY-155052-25
Verpackungseinheit
25 mg
Hersteller
MedChemExpress

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Product Description: PAD4-IN-2 (compound 5i) is a PAD4 inhibitor (IC50=1.94 μM). PAD4-IN-2 inhibits tumor growth in mice by specifically inhibiting the PAD4-H3cit-NETs pathway in neutrophils[1].

Applications: Cancer-programmed cell death

Formula: C20H23BClN7O6

References: [1]Zhu D, et al. Highly-tumor-targeted PAD4 inhibitors with PBA modification inhibit tumors in vivo by specifically inhibiting the PAD4-H3cit-NETs pathway in neutrophils. Eur J Med Chem. 2023 Oct 5;258:115619.

CAS Number: 2642327-52-2

Molecular Weight: 503.70

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Protein Arginine Deiminase
Mehr Informationen
Artikelnummer MEXHY-155052-25
Hersteller MedChemExpress
Hersteller Artikelnummer HY-155052-25
Green Labware Nein
Verpackungseinheit 25 mg
Mengeneinheit STK
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