RN-1665, CAS 1803003-65-7

Product Description: RN-1665 is an orally active TRPV4 antagonist that exhibits excellent selectivity for related TRP receptors such as TRPV1, TRPV3 and TRPM8. RN-1665 is a TRPV4 probe for focus screens, with IC50s of 0.26 μM and 0.39 μM for hTRPV4 and rTRPV4 from human and rat, respectively[1].

Applications: Neuroscience-Neuromodulation

Formula: C20H24F5N3O3S2

References: [1]Wei ZL, et al. Identification of orally-bioavailable antagonists of the TRPV4 ion-channel. Bioorg Med Chem Lett. 2015 Sep 15;25(18):4011-5.

CAS Number: 1803003-65-7

Molecular Weight: 513.54

Research Area: Others

Target: TRP Channel

• Artikelnummer: MEXHY-160900-0
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-160900-0
• Green Labware: Nein
• Verpackungseinheit: Get quote
• Mengeneinheit: STK