WNTinib, CAS 2770091-44-4

WNTinib, CAS 2770091-44-4
Artikelnummer
MEXHY-160765-25
Verpackungseinheit
25 mg
Hersteller
MedChemExpress

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Product Description: WNTinib (APS-8-100-2) is a multi-kinase inhibitor that selectively antagonizes β-catenin (CTNNB1) mutated hepatocellular carcinoma (HCC). WNTinib downregulates oncogenicWntsignaling by inhibiting KIT/MAPK and downstream EZH2 activation[1].

Applications: Cancer-Kinase/protease

Formula: C22H16F6N4O3

References: [1]Rialdi A, et al. WNTinib is a multi-kinase inhibitor with specificity against β-catenin mutant hepatocellular carcinoma. Nat Cancer. 2023 Aug;4(8):1157-1175.

CAS Number: 2770091-44-4

Molecular Weight: 498.38

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Apoptosis;Wnt
Mehr Informationen
Artikelnummer MEXHY-160765-25
Hersteller MedChemExpress
Hersteller Artikelnummer HY-160765-25
Green Labware Nein
Verpackungseinheit 25 mg
Mengeneinheit STK
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