INCB 13739, CAS 872506-67-7

Formulation: A solid

Formal Name: (3S)-1-[(3-chloro-2-methylphenyl)sulfonyl]-N-cyclohexyl-3-piperidinecarboxamide

Purity: ≥98%

Formula Markup: C19H27ClN2O3S

Formula Weight: 398,9

Shelf life (days): 1460

CAS Number: 872506-67-7

Notes: INCB 13739 is an inhibitor of 11β-hydroxysteroid dehydrogenase 1 (11β-HSD1; IC50 = 3.2 nM).{72228} It is greater than 1,000-fold selective for 11β-HSD1 over 11β-HSD2, the mineralocorticoid receptor, and the glucocorticoid receptor at 5 µM. INCB 13739 inhibits 11β-HSD1 activity in peripheral blood mononuclear cells (PBMCs; IC50 = 1.1 nM).

• Artikelnummer: CAY40223-50
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 40223-50
• Verpackungseinheit: 50 mg
• Mengeneinheit: STK