VCP-Eribulin, CAS 2130869-17-7

VCP-Eribulin, CAS 2130869-17-7
SKU
MEXHY-128871-0
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MedChemExpress

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Product Description: VCP-Eribulin consists the ADCs linker (VCP) and Eribulin[1]. Eribulin is a mechanistically unique microtubule inhibitor for cancer[2]. VCP-Eribulin is an Eribulin-based agent for antibody conjugates[1].

Applications: Cancer-programmed cell death

Formula: C59H86N6O16

References: [1]Earl F Albone, et al. Eribulin-based antibody-drug conjugates and methods of use. US20170252458A1./[2]Towle MJ, et al. Eribulin induces irreversible mitotic blockade: implications of cell-based pharmacodynamics for in vivo efficacy under intermittent dosing conditions. Cancer Res. 2011 Jan 15;71(2):496-505.

CAS Number: 2130869-17-7

Molecular Weight: 1135.34

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Drug-Linker Conjugates for ADC
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SKU MEXHY-128871-0
Manufacturer MedChemExpress
Manufacturer SKU HY-128871-0
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