Falnidamol, CAS 196612-93-8

Description: Falnidamol (BIBX 1382) is an orally active, selective EGFR tyrosine kinase inhibitor with an IC50 of 3 nM. It displays >1000-fold lower potency against ErbB2 (IC50=3.4 μM) and other related tyrosine kinases (IC50>10 μM). Falnidamol is a pyrimido-pyrimidine compound and exhibits anti-cancer activity.

CAS Number: 196612-93-8

Formula: C18H19ClFN7

Molecular Weight: 387,84

References: Solca FF, et al. Inhibition of epidermal growth factor receptor activity by two pyrimidopyrimidine derivatives. J Pharmacol Exp Ther. 2004 Nov;311(2):502-9.

• SKU: TGMTQ0271-2mg
• Manufacturer: TargetMol Chemicals
• Manufacturer SKU: TQ0271-2mg
• Package Unit: 2 mg
• Quantity Unit: STK