Product Description: Firsocostat (ND-630; GS-0976; NDI-010976) is an acetyl-CoA carboxylase (ACC) inhibitor; inhibits human ACC1 and ACC2 with IC50 values of 2.1 and 6.1 nM, respectively.
Applications: Metabolism-sugar/lipid metabolism
Formula: C28H31N3O8S
References: [1]Harriman G, et al. Acetyl-CoA carboxylase inhibition by ND-630 reduces hepatic steatosis, improves insulin sensitivity, and modulates dyslipidemia in rats. Proc Natl Acad Sci U S A. 2016 Mar 29;113(13):E1796-805.
CAS Number: 1434635-54-7
Molecular Weight: 569.63
Compound Purity: 99.96
Research Area: Metabolic Disease
Solubility: DMSO : ≥ 50 mg/mL
Target: Acetyl-CoA Carboxylase