GSK-6853, CAS 1910124-24-1

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CAS Number: 1910124-24-1

Description: GSK-6853 is a potent and selective BRPF1 inhibitor. GSK-6853 exhibits >1600-fold selectivity for BRPF1 over other bromodomains (pIC₅₀ values by TR-FRET are 8.1, 5.1/4.8 and 4.7/<4.3 for BRPF1, BRPF2/3 and BRD4 BD1/2, respectively). The structural analog of GSK-6853, GSK-9311, serves as a good inactive control (125- and 185-fold reduced potency in cell-free and cell-based assays, respectively).

Format: Solid

Storage Stability: At least 6 months at -20°C. 

Warnings: Avoid freeze/thaw cycles

Biosafety Level: Not applicable (BSL-1)

• SKU: BPS82067
• Manufacturer: BPS Bioscience
• Manufacturer SKU: 82067
• Package Unit: 50 mg
• Quantity Unit: STK