Product Description: GSK137647A (GSK 137647) is a potent, selective free fatty acid receptor 4 (FFA4) agonist with pEC50 values of 6.3, 6.2, and 6.1 for human, mouse and rat FFA4, and pEC50 values [1][2].
Applications: Metabolism-sugar/lipid metabolism
Formula: C16H19NO3S
References: [1]Salaga M, et, al. Activation of Free Fatty Acid Receptor 4 Affects Intestinal Inflammation and Improves Colon Permeability in Mice. Nutrients. 2021 Aug 6;13(8):2716. /[2]Sparks SM, et, al. Identification of diarylsulfonamides as agonists of the free fatty acid receptor 4 (FFA4/GPR120). Bioorg Med Chem Lett. 2014 Jul 15;24(14):3100-3.
CAS Number: 349085-82-1
Molecular Weight: 305.39
Compound Purity: 99.81
Research Area: Metabolic Disease
Solubility: DMSO : ≥ 100 mg/mL
Target: Free Fatty Acid Receptor