Formulation: A solid
Formal Name: 2-[(5-chloro-8-quinolinyl)oxy]-acetic acid, ethyl ester
Purity: ≥98%
Formula Markup: C13H12ClNO3
Formula Weight: 265,7
Shelf life (days): 1460
CAS Number: 88349-90-0
Notes: A2793 is an inhibitor of the two-pore domain potassium channel K2P18.1/TRESK (IC50 = 6.8 µM in ionomycin-stimulated Xenopus oocytes expressing the mouse receptor).{65336} It is selective for K2P18.1/TRESK over K2P2.1/TREK1, K2P10.1/TREK2, K2P4.1/TRAAK, K2P3.2/TASK2, K2P3.3/TASK3, K2P16.1/TALK1, and K2P13.1/THIK1 at 100 µM but does inhibit K2P3.1/TASK1.