Erlotinib-d6, CAS 1034651-23-4

Product Description: Erlotinib-d6 (CP-358774 D6) is a deuterium labeled Erlotinib (CP-358774). Erlotinib is a directly acting inhibitor EGFR tyrosine kinase inhibitor with an IC50 of 2 nM for human EGFR[1]. Erlotinib-d6 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

Applications: Cancer-Kinase/protease

Formula: C22H17D6N3O4

References: [1]Moyer JD, et al. Induction of apoptosis and cell cycle arrest by CP-358,774, an inhibitor of epidermal growth factor receptor tyrosine kinase. Cancer Res. 1997, 57(21), 4838-4848.

CAS Number: 1034651-23-4

Molecular Weight: 399.47

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: EGFR

• SKU: MEXHY-50896S-5
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-50896S-5
• Package Unit: 5 mg
• Quantity Unit: STK