N-Desmethyl apalutamide-d4

Product Description: N-Desmethyl apalutamide-d4 is the deuterium-labeled N-Desmethyl-Apalutamide (HY-135331). N-Desmethyl Apalutamide is an active metabolite of Apalutamide. N-Desmethyl Apalutamide is a less potent antagonist of the androgen receptor and is responsible for one-third of the activity of Apalutamide. The formation of N-Desmethyl Apalutamide mediated predominantly by CYP2C8 and CYP3A4. N-Desmethyl Apalutamide is moderate to strong CYP3A4 and CYP2B6 inducer and has an excellent plasma-proteins bound concentration[1][2][3].

Formula: C20H9D4F4N5O2S

Molecular Weight: 467.43

Compound Purity: 99.63

Research Area: Others

Solubility: 10 mM in DMSO

Target: Isotope-Labeled Compounds

• SKU: MEXHY-W754151-1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-W754151-1
• Green Labware: No
• Package Unit: 1 mg
• Quantity Unit: STK