2-chloro-N6-Cyclopentyladenosine (hydrate), CAS 1217443-91-8

Formulation: A crystalline solid

Formal Name: 2-chloro-N-cyclopentyl-adenosine, hemihydrate

Purity: ≥98%

Formula Markup: C15H20ClN5O4 • 0.5H2O

Formula Weight: 378,8

Shelf life (days): 1460

CAS Number: 1217443-91-8

Notes: 2-chloro-N6-Cyclopentyladenosine is an adenosine receptor agonist.{52004} It binds selectively to adenosine A1 receptors over A2A and A3 receptors with Ki values of 0.83, 2,300 and 42 nM, respectively, for the human recombinant receptors expressed in CHO cells. 2-chloro-N6-Cyclopentyladenosine decreases heart rate in isolated rat atria (EC50 = 8.2 nM) but does not affect vasodilation in bovine coronary arteries.{52005} It inhibits convulsions induced by isoniazid (Item No. 20378) and pentylenetetrazole (Item No. 18682) in mice when administered at a dose of 8.3 μmol/kg.{52006}

• SKU: CAY28731-50
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 28731-50
• Green Labware: No
• Package Unit: 50 mg
• Quantity Unit: STK