Formulation: A solid
Formal Name: 4-[(3R)-3-amino-1-pyrrolidinyl]-6,7-dihydro-5H-benzo[6,7]cyclohepta[1,2-d]pyrimidin-2-amine, dihydrochloride, hydrate
Purity: ≥98%
Formula Markup: C17H21N5 • 2HCl [XH2O]
Formula Weight: 368,3
Shelf life (days): 1460
Notes: A-943931 is a histamine H4 receptor antagonist (Ki = 3.8 nM).{57750} In vivo, A-943931 inhibits scratching induced by clobenpropit (Item No. 10011126) in mice (ED50 = 26 µmoles/kg, i.p.).