Formulation: A solid
Formal Name: 1-[10-[3-[4-(2-hydroxyethyl)-1-piperazinyl]propyl]-10H-phenothiazin-2-yl]-ethanone, dimaleate
Purity: ≥98%
Formula Markup: C23H29N3O2S • 2C4H4O4
Formula Weight: 643,7
Shelf life (days): 1460
CAS Number: 5714-00-1
Notes: Acetophenazine is a typical antipsychotic that binds to the serotonin (5-HT) receptor subtypes 5-HT6 and 5-HT7 and the androgen receptor (Kis = 72, 2.4, and 800 nM, respectively).{42535,54949} Acetophenazine also inhibits the binding of the sigma receptor agonist SKF 10047 (Ki = 36 nM) and the dopamine D2-selective antagonist spiperone (IC50 = 17 nM) to guinea pig brain membranes.{63241} It increases the duration of fighting and the latency to submission in mice.{63242}