Formulation: A solid
Formal Name: N-[[4-chloro-2-(1-methylethoxy)phenyl]methyl]-5-phenyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
Purity: ≥98%
Formula Markup: C21H20ClN5O
Formula Weight: 393,9
Shelf life (days): 1460
CAS Number: 1637300-25-4
Notes: AF64394 is an inverse agonist of the orphan G protein-coupled receptor GPR3.{62797} It selectively inhibits cAMP accumulation in HEK293 cells expressing GPR3 over GPR6 or GPR12 (IC50s = 0.5, 7.9, and 12 µM, respectively).