Formulation: A solid
Formal Name: 8-chloro-5,6-dihydro-5-methyl-1-[trans-4-(2-pyridinyloxy)cyclohexyl]-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine
Purity: ≥98%
Formula Markup: C22H24ClN5O
Formula Weight: 409,9
Shelf life (days): 1460
CAS Number: 1228088-30-9
Notes: Balovaptan is an antagonist of the vasopressin V1A receptors (Ki = 0.4 nM for the human receptor).{72076} It is selective for V1A receptors over V1B and V2 receptors and oxytocin (OT) receptors (Kis = >6,300, 2,474, and 1,063 nM, respectively, for the human receptors).