Bifeprunox (mesylate), CAS 350992-13-1

Formulation: A crystalline solid

Formal Name: 7-[4-([1,1′-biphenyl]-3-ylmethyl)-1-piperazinyl]-2(3H)-benzoxazolone, monomethanesulfonate

Purity: ≥98%

Formula Markup: C24H23N3O2 • CH3SO3H

Formula Weight: 481,6

Shelf life (days): 1460

CAS Number: 350992-13-1

Notes: Bifeprunox is an atypical antipsychotic.{52217} It is a dopamine D2 receptor partial agonist and an agonist of the serotonin (5-HT) receptor subtype 5-HT1A (Kis = 2.2 and 9.3 nM, respectively).{52219,52218} Bifeprunox inhibits apomorphine-induced climbing behavior in mice (ED50 = 0.1 mg/kg) and the conditioned avoidance response in rats (ED50 = 0.8 mg/kg).{52218} It decreases basal prepulse inhibition of the acoustic startle response in rats by 42% when administered at a dose of 10 mg/kg.{52219}

• SKU: CAY29523-10
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 29523-10
• Green Labware: No
• Package Unit: 10 mg
• Quantity Unit: STK