BMS 986187, CAS 684238-37-7

Formulation: A crystalline solid

Formal Name: 3,4,5,6,7,9-hexahydro-3,3,6,6-tetramethyl-9-[4-[(2-methylphenyl)methoxy]phenyl]-1H-xanthene-1,8(2H)-dione

Purity: ≥98%

Formula Markup: C31H34O4

Formula Weight: 470,6

Shelf life (days): 730

CAS Number: 684238-37-7

Notes: BMS 986187 is a positive allosteric modulator of δ-opioid receptors.{38565} In the presence of the endogenous δ-opioid receptor agonist leu-enkephalin, BMS 986187 has an average EC50 value of 30 nM for β-arrestin recruitment, but has little to no activity in the absence of an agonist. It is 100-fold selective for δ- over µ-opioid receptors in the presence of leu-enkephalin and the endogenous µ-opioid receptor agonist endomorphin I, respectively.

• SKU: CAY21549-10
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 21549-10
• Green Labware: No
• Package Unit: 10 mg
• Quantity Unit: STK