Formulation: A crystalline solid
Formal Name: 9-[4-[(2-bromophenyl)methoxy]phenyl]-3,4,5,6,7,9-hexahydro-3,3,6,6-tetramethyl-1H-xanthene-1,8(2H)-dione
Purity: ≥98%
Formula Markup: C30H31BrO4
Formula Weight: 535,5
Shelf life (days): 1460
CAS Number: 1776115-10-6
Notes: BMS 986188 is a positive allosteric modulator of δ-opioid receptors, with an EC50 value of 0.05 μM in a β-arrestin recruitment assay in the presence, but not absence, of the opioid receptor agonist leu-enkephalin (Item No. 23283).{38565} It is selective for δ- over μ-opioid receptors (EC50 = >10 μM) in the presence of leu-enkephalin and the μ-opioid receptor agonist endomorphin 1 (Item No. 23280), respectively.