Formulation: A solid
Formal Name: N-[2,6-dibromo-4-(1-methylethyl)phenyl]-N′-3-pyridinyl-urea
Purity: ≥98%
Formula Markup: C15H15Br2N3O
Formula Weight: 413,1
Shelf life (days): 1460
CAS Number: 688309-70-8
Notes: BX-430 is a noncompetitive allosteric antagonist of the purinergic P2X4 receptor (IC50s = 0.54 and 1.89 µM for the human and Xenopus receptors, respectively).{61154} BX-430 is selective for the human P2X4 receptor over the human P2X1, P2X2, P2X5, P2X3, and P2X7 receptors at 5 µM and over mouse and rat P2X4 receptors at 10 µM.